GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor gamma (ERRgamma) with an IC50 of 79 nM. GSK5182 does not interact with other nuclear receptors, including ERRalpha or ERalpha. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma (HCC)[1][2][3].
Molecular Weight:
417.55
Purity:
99.10
CAS Number:
[877387-37-6]
Formula:
C27H31NO3
Target:
Estrogen Receptor/ERR,Reactive Oxygen Species (ROS)
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted
