(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor gamma (ERRgamma) with an IC50 of 79 nM[1]. GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma[1][2][3].
Molecular Weight:
417.54
Purity:
98.90
CAS Number:
[2699724-40-6]
Formula:
C27H31NO3
Target:
Estrogen Receptor/ERR,Reactive Oxygen Species (ROS)
Application Notes:
MCE Product type: Reference compound
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