SGC-iMLLT is a first-in-class chemical probe and a potent, selective inhibitor of MLLT1/3-histone interactions with an IC50 of 0.26 µM. SGC-iMLLT shows high binding activity towards MLLT1 YEATS domain (YD) and MLLT3 YD (AF9/YEATS3) with Kds of 0.129 and 0.077 µM, respectively[1].
Molecular Weight:
388.47
Purity:
99.33
CAS Number:
[2255338-25-9]
Formula:
C22H24N6O
Target:
Epigenetic Reader Domain
Application Notes:
MCE Product type: Reference compound1
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