ERK-IN-4 is an ERK inhibitor binds preferentially to ERK2 with a Kd of 5 µM. ERK-IN-4 specificity inhibits ERK Rsk-1 and Elk-1 phosphorylation. ERK-IN-4 has little effect on ERK protein phosphorylation by its upstream activator MEK1/2[1].
Molecular Weight:
328.81
Purity:
98.30
CAS Number:
[1049738-54-6]
Formula:
C14H17ClN2O3S
Target:
ERK
Application Notes:
MCE Product type: Reference compound
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