BI-671800 is a highly specific and potent antagonist of chemoattractant receptor-homologous molecule on Th2 cells (DP2/CRTH2), with IC50 values of 4.5 nM and 3.7 nM for PGD2 binding to CRTH2 in hCRTH2 and mCRTH2 transfected cells, respectively[1]. BI-671800 has potential for the treatment of poorly controlled asthma[2].
Molecular Weight:
501.50
Purity:
99.36
CAS Number:
[1093108-50-9]
Formula:
C25H26F3N5O3
Target:
CRTH2 (GPR44),Prostaglandin Receptor
Application Notes:
MCE Product type: Reference compound
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