Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.
Molecular Weight:
618.47
Purity:
98.09
CAS Number:
[2247127-79-1]
Formula:
C26H24F3N7O3Se
Target:
Glutaminase
Application Notes:
Reference compound
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