A-953227 is a highly potent and selective inhibitor with the activity of inhibiting calcium-dependent esterase (calpain). A-953227 has enhanced selectivity for related cysteine proteases (cathepsins) and has shown good efficacy in cell experiments. A-953227 has shown broad efficacy in preclinical models for Alzheimers disease, suggesting that it has potential benefits in inhibiting Alzheimers disease[1].
Molecular Weight:
457.46
CAS Number:
[1037826-77-9]
Formula:
C25H20FN5O3
Target:
Ser/Thr Protease
Application Notes:
MCE Product type: Reference compound
* VAT and and shipping costs not included. Errors and price changes excepted
