R214127 is a selective mGlu1 receptor antagonist with IC50 values of 6 and 14 nM for rat and human mGlu1a. R214127 acts on a site from the glutamate binding pocket, and competes for the same transmembrane segment VII as other noncompetitive mGlu1 antagonists[1].
Molecular Weight:
303.35
CAS Number:
[409345-76-2]
Formula:
C20H17NO2
Target:
mGluR
Application Notes:
MCE Product type: Reference compound
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