BMS-470539 dihydrochloride is a highly potent and selective melanocortin-1 receptor (MC-1R) agonist with an IC50 of 120 nM, an EC50 of 28 nM. BMS-470539 dihydrochloride does not activate MC-3R and is a very weak partial agonist at MC-4R and MC-5R. BMS-470539 dihydrochloride has potently anti-inflammatory properties[1][2][3].
Molecular Weight:
632.62
Purity:
99.85
CAS Number:
[2341796-82-3]
Formula:
C32H43Cl2N5O4
Target:
Melanocortin Receptor
Application Notes:
MCE Product type: Reference compound1
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