PD 168368 is a potent, competitive, and selective neuromedin B receptor (NMB-R) antagonist with the Ki of 15-45 nM[1]. PD 168368 is neuromedin B receptor (NMBR, IC50=96 nM) / gastrin-releasing peptide receptor (GRPR IC50=3500 nM) antagonist[2]. PD 168368 also is a mixed FPR1/FPR2/FPR3 agonist with EC50s of 0.57, 0.24, and 2.7 nM, respectively[3].
Molecular Weight:
554.64
Purity:
99
CAS Number:
[204066-82-0]
Formula:
C31H34N6O4
Target:
Bombesin Receptor
Application Notes:
MCE Product type: Reference compound1
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