RP-69758 is a potent and selective non-peptide cholecystokinin-B (CCKB)/gastrin receptor antagonist. RP-69758 exhibits >200-fold selectivity for CCKB over CCKA receptors. RP-69758 antagonizes CCK-8-induced neuronal firing in rat hippocampal slices. RP-69758 inhibits Pentagastrin (HY-A0261)-induced gastric acid secretion in the rat. RP-69758 can be used for neurological disorders and gastrointestinal disease research[1].
Molecular Weight:
474.51
CAS Number:
[138562-23-9]
Formula:
C26H26N4O5
Target:
Cholecystokinin Receptor
Application Notes:
MCE Product type: Reference compound
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