BayCysLT2, an isophthalic acid derivative, is a selective and potent cysteinyl leukotriene 2 (CysLT2) receptor antagonist with an IC50 value of 53 nM. BayCysLT2 inhibits calcium mobilization induced by leukotriene D4 in HEK293 cells expressing human CysLT2 receptors. BayCysLT2 reverses LTC4-induced increases in coronary artery perfusion pressure and decreases in contractility in isolated perfused guinea pig hearts[1][2].
Molecular Weight:
589.68
Purity:
97.7
CAS Number:
[712313-33-2]
Formula:
C34H39NO8
Target:
Leukotriene Receptor
Application Notes:
MCE Product type: Reference compound
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