A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM)[1].
Molecular Weight:
320.43
Purity:
99.92
CAS Number:
[726174-00-1]
Formula:
C20H24N4
Target:
Dopamine Receptor
Application Notes:
MCE Product type: Reference compound
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