CDK12-IN-E9 is a potent and selective covalent CDK12 inhibitor and a non-covalent CDK9 inhibitor, while avoiding ABC transporter-mediated efflux. CDK12-IN-E9 has weak binding ability to CDK7/CyclinH complex with an IC50> 1 µM[1].
Molecular Weight:
434.53
Purity:
99.71
CAS Number:
[2020052-55-3]
Formula:
C24H30N6O2
Target:
CDK
Application Notes:
MCE Product type: Reference compound1
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