LP-403812 is a high affinity proline transporter (PROT) inhibitor that produces dose-dependent inhibition of hPROT (IC50=0.11 µM, Ki=0.12 µM) and also inhibits the activity of mouse brain synaptosomal mPROT with the same potency (IC50=0.23 µM). LP-403812 can be used to study the function of PROT in the brain[1].
Molecular Weight:
494.65
CAS Number:
[1142050-84-7]
Formula:
C26H34N6O2S
Target:
Amino acid Transporter
Application Notes:
MCE Product type: Reference compound
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