PWZ-029 is a selective inverse agonist for 5 GABAA receptors. PWZ-029 is a benzodiazepine site ligand. PWZ-029 shows a weak but significant partial agonistic effect at 1- and 3-containing receptors. PWZ-029 significantly increases retention session latency in mouse fibroblast cells. PWZ-029 can improve object recognition in normal and scopolamine-treated rat model[1][2].
Molecular Weight:
291.73
CAS Number:
[164025-33-6]
Formula:
C14H14ClN3O2
Target:
GABA Receptor
Application Notes:
MCE Product type: Reference compound
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