PD-135666 is a dipeptide inhibitor of cholecystokinin B (CCK B) receptors, binding to CCK B receptors in mouse cerebral cortex with IC50 of 0.1 nM. Its enantiomer, PD-140548, preferentially binds to CCK A receptors with IC50 of 2.8 nM in rat pancreas. PD-135666 exhibits anxiolytic effects in animal models[1].
Molecular Weight:
557.68
CAS Number:
[134557-41-8]
Formula:
C33H39N3O5
Target:
Cholecystokinin Receptor
Application Notes:
MCE Product type: Reference compound
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