GMA-839 is a selective modulator of the gamma-aminobutyric acid A receptor (GABAA) with an IC50 value of 230 nM. GMA-839 exhibits potent anxiolytic-like activity, demonstrating significant dose-dependent anxiolytic effects in animal models, with an effective oral dose of 1.6 mg/kg. Significant increases in punished responding were observed in squirrel monkeys and pigeons. GMA-839 shows promise for research in the field of anxiolytics[1].
Molecular Weight:
388.46
CAS Number:
[162882-76-0]
Formula:
C21H31F3O3
Target:
GABA Receptor
Application Notes:
Reference compound
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