SKI2496, CAS [[1308378-95-1]] Preis auf Anfrage

Product Overview

• Article Name: SKI2496, CAS [[1308378-95-1]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-117982
• Supplier Catalog Number: HY-117982
• Alternative Catalog Number: MCE-HY-117982-1UNIT
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

SKI2496 is an orally active GnRH receptor antagonist (IC50: 0.25 nM for hGnRHR, 13.2 nM for monkey GnRHR, 279.2 nM for rat GnRHR). SKI2496 blocks Ca2+ flux with an IC50 value of 0.76 nM. SKI2496 inhibits ERK1/2 phosphorylation with an IC50 value of 2.6 nM. SKI2496 inhbits serum LH concentrations, and can be used for research of sex hormone-dependent disorders[1].

Product Properties

• Molecular Weight: 739.68
• CAS Number: [1308378-95-1]
• Formula: C35H36F7N5O5
• Target: ERK,GnRH Receptor

Application Notes

• Application Notes: Reference compound