GSK466317A is a PKA inhibitor, with an IC50 of 12.59 µM. GSK466317A also inhibits GRK1, GRK2, and GRK5, with IC50s of 1000, 31.62, and 39.81 µM, respectively[1].
Molecular Weight:
448.83
CAS Number:
[864082-48-4]
Formula:
C21H16ClF3N4O2
Target:
G Protein-coupled Receptor Kinase (GRK),PKA
Application Notes:
MCE Product type: Reference compound
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