BRM/BRG1 ATP Inhibitor-1 (compound 14) is an orally active allosteric dual brahma homolog (BRM)/SWI/SNF related matrix associated actin dependent regulator of chromatin subfamily A member 2 (SMARCA2) and brahma related gene 1 (BRG1)/SMARCA4 ATPase activity inhibitor, both IC50s are below 0.005 µM. BRM/BRG1 ATP Inhibitor-1 has anticancer activity[1].
Molecular Weight:
318.27
Purity:
99.72
CAS Number:
[2270879-17-7]
Formula:
C11H9F3N4O2S
Target:
Epigenetic Reader Domain
Application Notes:
MCE Product type: Reference compound
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