9-Ethyladenine is a precursor of competitive antagonists of adenosine receptors (A1, A2, A3), with no significant inhibitory effect on adenine phosphoribosyltransferase (APRT). 9-Ethyladenine derivatives have high affinity and selectivity for A1 (Ki=27 nM), A2A (Ki=46 nM), and A3 (Ki=86 nM) receptors. 9-Ethyladenine does not inhibit brain APRT activity, can be used in the study of adenosine receptor-related diseases (such as nervous system diseases) models[1][2].
Molecular Weight:
163.18
Purity:
99.87
CAS Number:
[2715-68-6]
Formula:
C7H9N5
Target:
Adenosine Receptor
Application Notes:
MCE Product type: Natural Products
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