VU0467485, CAS [[1451994-10-7]]

Product Overview

• Article Name: VU0467485, CAS [[1451994-10-7]]
• Biozol Catalog Number: MCE-HY-120184
• Supplier Catalog Number: HY-120184
• Alternative Catalog Number: MCE-HY-120184-10MG,MCE-HY-120184-25MG,MCE-HY-120184-10MMX1ML,MCE-HY-120184-100MG,MCE-HY-120184-5MG,MCE-HY-120184-50MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: AZ13713945

Product Description

VU0467485 (AZ13713945) is a potent, selective, and orally bioavailable muscarinic acetylcholine receptor 4 (M4) positive allosteric modulator (PAM). VU0467485 (AZ13713945) potentiates activity of ACh at M4 with EC50s of 26.6 nM and 78.8 nM at rat and human M4 receptors, respectively. VU0467485 (AZ13713945) shows selectivity for M4 over human and rat M1/2/3/5. VU0467485 (AZ13713945) displays moderate to high CNS penetration. VU0467485 (AZ13713945) has antipsychotic-like activity[1].

Product Properties

• Molecular Weight: 360.41
• Purity: 99.29
• CAS Number: [1451994-10-7]
• Formula: C17H17FN4O2S
• Target: mAChR

Application Notes

• Application Notes: MCE Product type: Reference compound