VU0463841 is a potent, selective and brain-penetrant mGlu5 negative allosteric modulator (NAM) with an IC50 of 13 nM. VU0463841 is ineffective against mGlu1-4 and mGlu7-8. VU0463841 has the potential for the Cocaine addiction research[1].
Molecular Weight:
290.68
CAS Number:
[1439095-16-5]
Formula:
C13H8ClFN4O
Target:
mGluR
Application Notes:
MCE Product type: Reference compound
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