BMS-986187 is an delta-opioid receptor-selective positive allosteric modulator (PAM) with an EC50 of 0.03 µM and a pKB of 6.02 (~1 µM). BMS-986187 has no observable PAM activity at the µ-receptor (EC50=3 µM)[1].
Molecular Weight:
470.60
Purity:
99.66
CAS Number:
[684238-37-7]
Formula:
C31H34O4
Target:
Opioid Receptor
Application Notes:
Reference compound
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