MRS 1523 is a potent and selective adenosine A3 receptor antagonist with Ki values of 18.9 nM and 113 nM for human and rat A3 receptors, respectively. In rat this corresponds to selectivities of 140- and 18-fold vs A1 and A2A receptors, respectively. MRS 1523 can exert antihyperalgesic effect through N-type Ca channel block and action potential inhibition in isolated rat dorsal root ganglion (DRG) neurons[1][2].
Molecular Weight:
399.55
Purity:
99.97
CAS Number:
[212329-37-8]
Formula:
C23H29NO3S
Target:
Adenosine Receptor,Calcium Channel
Application Notes:
MCE Product type: Reference compound
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