A778317 is a TRPV1 antagonists. A778317 can block changes in intracellular calcium levels mediated by TRPV1 receptors, with a pIC50 value of 8.31. A-778317 can also block the activation of natural rat TRPV1 receptors in dorsal root ganglion neurons by capsaicin and acid[1].
Molecular Weight:
359.46
CAS Number:
[808756-64-1]
Formula:
C23H25N3O
Target:
Others
Application Notes:
MCE Product type: Reference compound
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