Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist, inhibits [3H]SP binding to the NK1 receptor with pKi values of 9.5 and 10.6 in rat and human membranes respectively, acts as a potential broad-spectrum anti-emetic agent[1].
Molecular Weight:
505.36
Purity:
99.56
CAS Number:
[168266-51-1]
Formula:
C21H25Cl2F3N6O
Target:
Neurokinin Receptor
Application Notes:
MCE Product type: Reference compound1
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