KRH-3955 hydrochloride is an orally bioavailable CXCR4 antagonist. KRH-3955 hydrochloride inhibits SDF-1alpha binding to CXCR4 with an IC50 of 0.61 nM. KRH-3955 hydrochloride is also a highly potent and selective inhibitor of X4 HIV-1, with an EC50 of 0.3 to 1.0 nM[1].
Molecular Weight:
589.09
Purity:
97.50
CAS Number:
[2253744-59-9]
Formula:
C28H48Cl3N7
Target:
CXCR,HIV
Application Notes:
MCE Product type: Reference compound
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