Thioperamide maleate (MR-12842 maleate) is a potent, orally available, brain penetrant and selective H3 receptor antagonist with a Ki of 4.3 nM for inhibition of [3H]histamine release. Thioperamide maleate inhibits [3H]histamine synthesis with a Ki of 31 nM[1].
Purity:
98.26
CAS Number:
[148440-81-7]
Formula:
C15H24N4S.xC4H4O4
Target:
Histamine Receptor
Application Notes:
MCE Product type: Reference compound
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