A-317920 is a selective and potent rat histamine H3 receptor (H3R) antagonist with pKi value of 9.2 and 7.0 for full-length rat and full-length human H3R, respectively. A-317920 exhibits over 130 fold selective affinity for the rat over the human H3R. A-317920 enhances cognition via H3R blockade[1].
Molecular Weight:
453.53
CAS Number:
[360551-59-3]
Formula:
C25H31N3O5
Target:
Histamine Receptor
Application Notes:
MCE Product type: Reference compound
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