GBR 12935 is a potent, and selective dopamine reuptake inhibitor, with the binding constant (Kd) of 1.08 nM in COS-7 cells. GBR 12935 stimulates the locomotion activity in different mice strains but fails to induce stereotypy. Thus, GBR 12935 also prevents the d-Fenfluramine-induced head-twitch response in mice[1][2][3][4].
Molecular Weight:
414.58
CAS Number:
[76778-22-8]
Formula:
C28H34N2O
Target:
Dopamine Transporter
Application Notes:
MCE Product type: Reference compound
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