VU0134992 is the first subtype-preferring, orally active and selective Kir4.1 potassium channel pore blocker, with an IC50 of 0.97 µM. VU0134992 is 9-fold selective for homomeric Kir4.1 over Kir4.1/5.1 concatemeric channels (IC50=9 µM) at -120 mV[1].
Molecular Weight:
411.38
Purity:
99.30
CAS Number:
[755002-90-5]
Formula:
C20H31BrN2O2
Target:
Potassium Channel
Application Notes:
MCE Product type: Reference compound
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