CHMFL-KIT-031 is a highly selective KIT V559D inhibitor, with an IC50 of 28 nM. CHMFL-KIT-031 potently affects KIT V559D mutants phosphorylation at Y703/719/823 sites. CHMFL-KIT-031 inhibits the tumor growth in BaF3-TEL-KIT-V559D cell inoculated mouse model[1].
Molecular Weight:
487.51
Formula:
C26H25N5O5
Target:
c-Kit
Application Notes:
MCE Product type: Reference compound1
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