CVT-2759 is a potent inhibitor of A1-ADOR, with the IC50 values of 0.18 µM and 9.5 µM to reduce the binding of [3H]CPX in the absence and presence of 1 mM GTP. CVT-2759 plays an important role in slowing AV nodal conduction and thereby ventricular rate without causing AV block, bradycardia, atrial arrhythmias, or vasodilation[1].
Molecular Weight:
394.38
CAS Number:
[342419-09-4]
Formula:
C16H22N6O6
Target:
Adenosine Receptor
Application Notes:
MCE Product type: Reference compound
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