GSK484, a chemical probe, is a PAD4 inhibitor. GSK484 reduces inflammation and joint destruction in CIA mouse models. GSK484 inhibits TNF-alpha expression and reverses Erastin-induced gut dysbiosis. GSK484 can be used in rheumatoid arthritis (RA) research[1].
Molecular Weight:
473.57
Purity:
99.14
CAS Number:
[1652629-23-6]
Formula:
C27H31N5O3
Target:
Protein Arginine Deiminase
Application Notes:
MCE Product type: Reference compound
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