BQ-123 is a potent and selective endothelin A (ETA) receptor antagonist with an IC50 of 7.3 nM and a Ki of 25 nM. BQ-123 inhibits endothelin-1-mediated proliferation of human pulmonary artery smooth muscle cells and lowers blood pressure in different rat models of hypertension[1][2][3].
Molecular Weight:
610.70
Purity:
99.82
CAS Number:
[136553-81-6]
Formula:
C31H42N6O7
Target:
Endothelin Receptor
Application Notes:
MCE Product type: Reference compound
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