Stenoparib (E7449) is a potent PARP1 and PARP2 inhibitor and also inhibits TNKS1 and TNKS2, with IC50s of 2.0, 1.0, ~50 and ~50 nM for PARP1, PARP2, TNKS1 and TNKS2, respectively, using 32P-NAD+ as substrate.
Molecular Weight:
317.34
Purity:
98
CAS Number:
[1140964-99-3]
Formula:
C18H15N5O
Target:
PARP
Application Notes:
MCE Product type: Reference compound
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