HET0016 is a potent and selective 20-hydroxyeicosatetraenoic acid (20-HETE) synthase inhibitor, with IC50 values of 17.7 nM, 12.1 nM and 20.6 nM for recombinant CYP4A1-, CYP4A2- and CYP4A3-catalyzed 20-HETE synthesis, respectively. HET0016 also is a selective CYP450 inhibitor, which has been shown to inhibit angiogenesis and tumor growth[1][2].
Molecular Weight:
206.28
Purity:
99.69
CAS Number:
[339068-25-6]
Formula:
C12H18N2O
Target:
Cytochrome P450
Application Notes:
MCE Product type: Reference compound
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