TBK1/IKKepsilon-IN-4 is a 6-aminopyrazolopyrimidine derivative and a potent, selective TBK1 and IKKepsilon inhibitor with IC50 values of 13 nM and 59 nM, respectively. TBK1/IKKepsilon-IN-4 shows 100- to 1000-fold less activity against other protein kinases including PDK1, PI3K family members and mTOR[1].
Molecular Weight:
533.62
Purity:
99.42
CAS Number:
[1381930-17-1]
Formula:
C28H35N7O4
Target:
IKK
Application Notes:
MCE Product type: Reference compound
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