PU139 is a potent pan-histone acetyltransferase (HAT) inhibitor. PU139 blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB (cAMP response element-binding) protein (CBP) and p300 with IC50s of 8.39, 9.74, 2.49 and 5.35 µM, respectively[1][2].
Molecular Weight:
246.26
Purity:
99.51
CAS Number:
[158093-65-3]
Formula:
C12H7FN2OS
Target:
Histone Acetyltransferase
Application Notes:
MCE Product type: Reference compound
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