GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 also shows binding to RIPK2[1].
Molecular Weight:
370.40
Purity:
98.79
CAS Number:
[319492-82-5]
Formula:
C20H22N2O5
Target:
Cyclin G-associated Kinase (GAK)
Application Notes:
MCE Product type: Reference compound
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