Spiradoline mesylate (U-62066 mesylate), an arylacetamide, is a selective kappa opioid receptor (KOR) agonist with a Ki of 8.6 nM in guinea pig. The Ki values of Spiradoline mesylate for µ and delta receptors are 252 nM and 9400 nM, respectively. Spiradoline mesylate has potent diuretic, analgesic, antiarrythmic, antitussive, neuroprotective properties and easily penetrates the blood-brain barrier[1][2].
Molecular Weight:
521.50
Purity:
99.95
CAS Number:
[87173-97-5]
Formula:
C23H34Cl2N2O5S
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound
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