GV-58 is a novel N- and P/Q-type calcium (Ca2+) channel agonist with EC50s of 7.21 and 8.81 µM, respectively. GV-58 slows the deactivation of channels, resulting in a large increase in presynaptic Ca2+ entry during activity. GV-58 can be used in lambert-eaton myasthenic syndrome (LEMS) research[1][2][3].
Molecular Weight:
374.50
Purity:
99.22
CAS Number:
[1402821-41-3]
Formula:
C18H26N6OS
Target:
Calcium Channel
Application Notes:
MCE Product type: Reference compound1
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