(R)-OP-1074 is an isomer of OP-1074 (HY-125263) and can serve as a control compound in experiments. OP-1074, a pure anti-estrogen drug, is a selective ER degrader (PA-SERD) with specific anti-estrogenic activity against ERalpha and ERbeta, inhibiting 17beta-estradiol (E2)-stimulated transcription with IC50 values of 1.6 and 3.2 nM, respectively.
Molecular Weight:
457.56
Purity:
98.24
CAS Number:
[1443752-77-9]
Formula:
C29H31NO4
Target:
Estrogen Receptor/ERR
Application Notes:
MCE Product type: Reference compound
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