ES 6864 is an orally active, competitive inhibitor for human renin, with an IC50 of 6.9 nM and a Ki of 7.3 nM. ES 6864 exhibits high species-specific and enzyme-specific properties. ES 6864 exhibits metabolic stability in rat tissue homogenates. ES 6864 reduces blood pressure in rats and sodium-depleted awake marmosets[1].
Molecular Weight:
791.01
CAS Number:
[116326-39-7]
Formula:
C42H58N6O7S
Target:
Renin
Application Notes:
MCE Product type: Reference compound
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