ARC 239 dihydrochloride is a selective alpha2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at alpha2A, alpha2B, and alpha2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively[1].
Molecular Weight:
480.43
Purity:
99.20
CAS Number:
[55974-42-0]
Formula:
C24H31Cl2N3O3
Target:
Adrenergic Receptor
Application Notes:
MCE Product type: Reference compound
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