CARM1-IN-1 (hydrochloride), CAS [[2070018-31-2]]

Product Overview

• Article Name: CARM1-IN-1 (hydrochloride), CAS [[2070018-31-2]]
• Biozol Catalog Number: MCE-HY-12759A
• Supplier Catalog Number: HY-12759A
• Alternative Catalog Number: MCE-HY-12759A-10MG,MCE-HY-12759A-5MG,MCE-HY-12759A-25MG,MCE-HY-12759A-50MG,MCE-HY-12759A-100MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

CARM1-IN-1 (compound 7g) hydrochloride is a highly potent and selective inhibitor of CARM1 (IC50=8.6 µM, CARM1/PABP1), with low inhibitory activity against PRMT1 and SET7 (IC50 >667 µM). CARM1-IN-1 hydrochloride inhibits the methylation activity of CARM1 and the methylation levels of different substrates, such as PABP1, CA150, SmB, and H3. CARM1-IN-1 hydrochloride also inhibits the promoter activity of prostate-specific antigen (PSA) without significant cytotoxicity[1].

Product Properties

• Molecular Weight: 591.72
• Purity: 95.13
• CAS Number: [2070018-31-2]
• Formula: C26H22Br2ClNO3
• Target: Histone Methyltransferase

Application Notes

• Application Notes: MCE Product type: Reference compound