N-Desmethyl-loperamide is a major metabolite of loperamide, a drug that selectively activates peripheral µopioid receptors with a Ki value of 0.16 nM. N-Desmethyl-loperamide is a substrate of the ATP-dependent efflux transporter P-glycoprotein[1][2][3].
Molecular Weight:
463.01
Purity:
98.36
CAS Number:
[66164-07-6]
Formula:
C28H31ClN2O2
Target:
Opioid Receptor
Application Notes:
MCE Product type: Reference compound1
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