Pelabresib (CPI-0610) is a potent, selective, orally active and cell-active BET inhibitor. Pelabresib inhibits BRD4-BD1 with an IC50 of 39 nM, and with an EC50 value of 0.18 µM for MYC[1].
Molecular Weight:
365.81
Purity:
99.95
CAS Number:
[1380087-89-7]
Formula:
C20H16ClN3O2
Target:
Epigenetic Reader Domain
Application Notes:
Reference compound
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